Cabergoline (active ingredient) – suppresses the secretion of prolactin , besides it increases libido and erection significantly reduces recovery time between sexual acts, and also lowers blood pressure. Cabergoline relates to derivatives of ergot alkaloids, the mechanism of action – the agonist of dopamine (D2) receptors. It is more modern and safe analogue bromocriptine .
Formulation almost completely eliminates the major side effects of steroids such as the deck (Deck-dik) and Trenbolone . One of the effects caused by the decrease in prolactin kontsetratsii – decrease fluid retention in the tissues, which gives more gain in lean muscle mass.
Cabergoline is available in pharmacies under the trade names:
- Bergolak (700-900 rubles 8 tablets 0.5 mg). (In 2014, the manufacturer does not renew the license, as of January 2016. Production is not renewed, the management announced that production will be resumed in the summer of 2016 already appears in the sale).
- Agalates (1000-1450 rubles 8 tablets 0.5 mg).
- Dostinex (1600-3000 rubles per 8 tablets of 0.5 mg) – the original drug, which appeared on the market in 1985.
Prices are per 10/08/2015
- Cabergoline (700-900 rubles 8 tablets 0.5 mg)
- Dostinex (1700-1900 rubles 8 tablets 0.5 mg)
The mechanism of action
The main mechanism of action is the activation of the cabergoline D2 receptors that are located on laktotrofnyh pituitary cells. Stimulation of the dopamine receptors in this area leads to a decrease in the secretory function of cells producing prolactin.
In addition it was found interaction with other receptors: D3, D4, 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, α2B. Α2B receptor antagonism with further explains the beneficial effect on the erectile function (expansion corpus cavernosum occurs).
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Experience in the application showed that the optimal scheme to reduce the use of cabergoline prolactin constructed as follows:
- During the course of progestin anabolic steroids ( nandrolone , trenbolone ): 0.25 mg (. Whole or 1/2 tab) every 7-21 days, starting from the third or fourth week of the course, when the concentration of the ACC is close to the maximum. Optimum dosage and frequency of administration selected under control of prolactin level assays, since the effect of the drug differs depending on the individual.
- With increasing prolactin levels above the permissible reception frequency increases: 0.25 mg every 4 day. Control prolactin desirable to perform analysis after two techniques with subsequent correction circuit.
The drug is taken as a meal or on an empty stomach.
The study on 200 patients, Parkinson’s patients with high cabergoline doses (0.5 mg daily) reports on the following side effects:
- The digestive system (the most common): nausea , constipation , dry mouth, dyspepsia
- Nervous system: insomnia, dizziness, depression, distortion of consciousness
- Cardiovascular system: fall in blood pressure, peripheral edema, dysrhythmia, damage to valves, pericarditis
- Immune system: rarely – hypersensitivity reactions, skin rash.
- From hemopoiesis system: seldom – rodonalgia.
- The respiratory system: often – shortness of breath, rarely – pleural effusion, lung fibrosis, nasal bleeding.
If you are using low doses side effects are rare or completely absent. On the forums most commonly reported depressed mood and loss of appetite.
Do not take more often one tablet a week (with the exception – highly elevated levels of prolactin).
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